BDBM50396018 CHEMBL1230640

SMILES OC(=O)c1ccc(O)c2ncccc12

InChI Key InChIKey=JGRPKOGHYBAVMW-UHFFFAOYSA-N

Data  36 IC50  1 Kd  1 EC50

PDB links: 7 PDB IDs match this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50396018   

TargetMethylcytosine dioxygenase TET2(Homo sapiens)
Tu Dortmund University

Curated by ChEMBL
LigandPNGBDBM50396018(CHEMBL1230640)
Affinity DataIC50:  2.27E+3nMAssay Description:Inhibition of N-terminal His6-tagged TET2 (unknown origin) expressed in Escherichia coli assessed as reduction in hmC and fC levels preincubated for ...More data for this Ligand-Target Pair
In DepthDetails PubMed